Production Method 1

254454-54-1

2564-83-2

1765-93-1

2222044-40-6

398-23-2

1044507-64-3

Reaction Conditions

1.1R:(Me3Si)2NH ?Na, C:13462-90-3, C:5456-63-3, S:Me2CHOH, S:THF, 30 min, 80°C

Reference

Microwave-Assisted Suzuki-Miyaura Cross Coupling using Nickel as Catalyst to Rapidly Access to 3-Arylazetidine

By Dequirez, Geoffroy et al, ChemistrySelect, 2017, 2(28), 8841-8846

1-Azetidinecarboxylic acid, 3-[(2,2,6,6-tetramethyl-1-piperidinyl)oxy]-, 1,1-dimethylethyl ester Raw materials

• 1-Boc-3-iodoazetidine
• Tempo
• 4-Fluorobenzeneboronic acid

1-Azetidinecarboxylic acid, 3-[(2,2,6,6-tetramethyl-1-piperidinyl)oxy]-, 1,1-dimethylethyl ester Preparation Products

• 4,4'-Difluorobiphenyl (398-23-2)
• 1-Azetidinecarboxylic acid, 3-(4-fluorophenyl)-, 1,1-dimethylethyl ester (1044507-64-3)
• 1-Azetidinecarboxylic acid, 3-[(2,2,6,6-tetramethyl-1-piperidinyl)oxy]-, 1,1-dimethylethyl ester (2222044-40-6)

• 1. Exciplex emission from the mixed dimer of naphthalene and 2-cyanonaphthalene in a supersonic jet
  Aloke Das,K. K. Mahato,Chayan K. Nandi,Tapas Chakraborty,Shridhar R. Gadre,Nikhil A. Gokhale Phys. Chem. Chem. Phys., 2002,4, 2162-2168
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  Alexandre Vimont,Arnaud Travert,Philippe Bazin,Jean-Claude Lavalley,Marco Daturi,Christian Serre,Gérard Férey,Sandrine Bourrelly,Philip L. Llewellyn Chem. Commun., 2007, 3291-3293
• 4. Excellent electrochemical performance of LiFe0.4Mn0.6PO4 microspheres produced using a double carbon coating process?
  Yong Ping Huang,Tao Tao,Zheng Chen,Wei Han,Ying Wu,Chunjiang Kuang,Shaoxiong Zhou,Ying Chen J. Mater. Chem. A, 2014,2, 18831-18837
• 5. Fast-pulsing NMR techniques for the detection of weak interactions: successful natural abundance probe of hydrogen bonds in peptides?
  Amandine Altmayer-Henzien,Valérie Declerck,David J. Aitken,Ewen Lescop,Denis Merlet,Jonathan Farjon Org. Biomol. Chem., 2013,11, 7611-7615

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