Bioisosteric replacement of the pyrazole 3-carboxamide moiety of rimonabant. A novel series of oxadiazoles as CB1 cannabinoid receptor antagonists?
Organic & Biomolecular Chemistry Pub Date: 2008-07-23 DOI: 10.1039/B807648K
Abstract
Based on the bioisosteric replacement of the pyrazole C3-carboxamide of rimonabant with a 5-alkyl oxadiazole ring, a novel class of
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Journal Name：Organic & Biomolecular Chemistry
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CAS no.: 89640-58-4
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