Diversity oriented synthesis of 6-nitro- and 6-aminoquinolones and their activity as alkaline phosphatase inhibitors?
RSC Advances Pub Date: 2015-07-06 DOI: 10.1039/C5RA10948E
Abstract
The novel quinolone derivatives synthesized by cyclization of α,β-ynones with primary amines were shown to be promising TNAP and IAP inhibitors. The mechanism of their formation was studied by the isolation of intermediates.
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Journal Name：RSC Advances
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CAS no.: 89640-58-4
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