Production Method 1

117098-94-9

2824235-75-6

Reaction Conditions

1.1 Reagents: Diisopropylethylamine Catalysts: 4-(Dimethylamino)pyridine Solvents: Dichloromethane ;  0 °C → rt; overnight, rt

Reference

Discovery of potent benzoxaborole inhibitors against SARS-CoV-2 main and dengue virus proteases

Kuehl, Nikos; Lang, Johannes; Leuthold, Mila M.; Klein, Christian D., European Journal of Medicinal Chemistry, 2022, 240,

benzyl N-(1-hydroxy-1,3-dihydro-2,1-benzoxaborol-6-yl)carbamate Raw materials

• 5-Aminoboronphthalide

benzyl N-(1-hydroxy-1,3-dihydro-2,1-benzoxaborol-6-yl)carbamate Preparation Products

• benzyl N-(1-hydroxy-1,3-dihydro-2,1-benzoxaborol-6-yl)carbamate (2824235-75-6)

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