Br?nsted acid cocatalysis in photocatalytic intramolecular coupling of tertiary amines: efficient synthesis of 2-arylindols?
Organic & Biomolecular Chemistry Pub Date: 2016-07-11 DOI: 10.1039/C6OB01239F
Abstract
We report herein a highly efficient intramolecular coupling reaction of tertiary amines and ketones (α,β-unsaturated ketones) by using a Br?nsted acid as a cocatalyst, affording 2-arylindols in good to excellent yields (up to 92%) under visible light irradiation at room temperature.
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Journal Name：Organic & Biomolecular Chemistry
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CAS no.: 89640-58-4
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