Design and synthesis of β-amino alcohol based β-lactam–isatin chimeras and preliminary analysis of in vitro activity against the protozoal pathogen Trichomonas vaginalis?
MedChemComm Pub Date: 2013-04-16 DOI: 10.1039/C3MD00057E
Abstract
We have described the synthesis of β-amino alcohol based β-lactam–isatin chimeras along with their in vitro evaluation against T. vaginalis. SAR studies showed dependence of activity on concentration as well as substituent on N-1 of β-lactam and C-5 of
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Journal Name：MedChemComm
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CAS no.: 89640-58-4
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