Synthesis of acridines via copper-catalyzed amination/annulation cascades between arylboronic acids and anthranils?
Organic & Biomolecular Chemistry Pub Date: 2022-11-23 DOI: 10.1039/D2OB01705A
Abstract
Copper-catalyzed tandem cyclization reactions between arylboronic acids and anthranils have been established, providing new approaches for one-pot assembly of azacycle acridines. This one-pot protocol features simple operation, precious-metal-free conditions and good functional group compatibility, thus providing an efficient approach for the synthesis of a variety of acridines in moderate to good yields.
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Journal Name：Organic & Biomolecular Chemistry
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CAS no.: 89640-58-4
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