Organocatalytic asymmetric synthesis of arylindolyl indolin-3-ones with both axial and central chirality?
Chemical Communications Pub Date: 2020-09-11 DOI: 10.1039/D0CC05432A
Abstract
An efficient method for chiral phosphoric acid-catalyzed asymmetric synthesis of arylindolyl indolin-3-ones with both axial and central chirality has been developed via the reaction of 3-arylindoles with 2-aryl-3H-indol-3-ones, and the target products were obtained in high yields with excellent enantioselectivity and diastereoselectivity.
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Journal Name：Chemical Communications
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CAS no.: 89640-58-4
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