Formal synthesis of (+)-lactacystin from l-serine?
RSC Advances Pub Date: 2019-09-24 DOI: 10.1039/C9RA07244F
Abstract
A formal, stereocontrolled synthesis of lactacystin has been completed from t-Bu-O-L-serine, providing the key intermediate 13, also useful for the generation of a range of C-9 analogues.
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Journal Name：RSC Advances
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CAS no.: 89640-58-4
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