Benzazocines
Benzazocines are a class of chemical compounds characterized by a benzene ring fused to an azocine ring, which is itself formed from two pyrrole rings. These drugs possess analgesic and anti-inflammatory properties due to their structural similarity to the endogenous opioids. Benzazocines act as partial agonists at mu-opioid receptors, providing moderate pain relief without the severe side effects often associated with full opioid agonists such as morphine or fentanyl. They are also used in veterinary medicine for pain management. Common examples include pentazocine and butorphanol, which have a lower risk of causing respiratory depression compared to traditional opioids. Due to their potential for abuse, benzazocines are typically prescribed under strict medical supervision.
| Structure | Chemical Name | CAS | MF |
|---|---|---|---|
![]() |
Saframycin R | 85411-35-4 | C31H34N4O10 |
![]() |
Cenicriviroc | 497223-25-3 | C41H52N4O4S |
![]() |
Propanamide,N-[[(6R,7R,9R,14aS,15R)-7-cyano-6,7,9,10,13,14,14a,15-octahydro-1,4-dihydroxy-2,11-dimethoxy-3,12,16-trimethyl-5,10,13-trioxo-6,15-imino-5H-isoquino[3,2-b][3]benzazocin-9-yl]methyl]-2-oxo- | 92569-03-4 | C29H30N4O9 |
![]() |
ecteinascidin 770 S-oxide | 442851-31-2 | C40H42N4O11S |
![]() |
2,5-Ethano-2H-azocino[4,3-b]indole,4-ethylidene-1,3,4,5,6,7-hexahydro-6-methylene-, (4E,5R)- | 3463-93-2 | C18H20N2 |
![]() |
Ecteinascidin 770 | 114899-80-8 | C40H42N4O10S |
![]() |
Indeno[1,2-c]pyrrole-6,7-diol,1,2,3,3a,8,8a-hexahydro-2-methyl- | 103810-34-0 | C12H15NO2 |
![]() |
Saframycin D | 66082-30-2 | C28H31N3O9 |
![]() |
Saframycin E | 66082-31-3 | C28H33N3O9 |
![]() |
(3AR*,8R*,8aR*)-tert-Butyl 8-amino-3,3a,8,8atetra-hydroindeno2,1-cpyrrole-2(1H)-carboxylate | 1251007-19-8 | C16H22N2O2 |
Related Literature
-
Michael Kappl,Paul M. Young,Daniela Traini,Sanyog Jain RSC Adv., 2016,6, 25789-25798
-
Li-Hua Gan,Rui Wu,Jian-Lei Tian,Patrick W. Fowler Phys. Chem. Chem. Phys., 2017,19, 419-425
-
Chongyang Zhu,Xiaojia Bian,Xin Jia,Ning Tang,Yongqiang Cheng Food Funct., 2020,11, 10635-10644
-
Yuan-Jun Tong,Lu-Dan Yu,Lu-Lu Wu,Shu-Ping Cao,Ru-Ping Liang,Li Zhang,Xing-Hua Xia,Jian-Ding Qiu Chem. Commun., 2018,54, 7487-7490
-
M. Sheykhan,S. Khani,S. Shaabanzadeh,M. Joafshan Green Chem., 2017,19, 5940-5948
Recommended suppliers
-
Wuhan Comings Biotechnology Co., Ltd.Factory Trade Brand reagentsCompany nature: Private enterprises
-
Beyond Pharmaceutical Co., LtdFactory Trade Brand reagentsCompany nature: Private enterprises
-
HANGZHOU BAIS CHEMICAL TECHNOLOGY CO., LTD.Factory Trade Brand reagentsCompany nature: Private enterprises
-
Tiancheng Chemical (Jiangsu) Co., LtdFactory Trade Brand reagentsCompany nature: Private enterprises
-
Shanghai Jinhuan Chemical CO., LTD.Factory Trade Brand reagentsCompany nature: Private enterprises
Recommended products









